Labetalol 100mg

Generic For: Trandate

Labetalol 100mg (brand name Trandate) is a combined alpha- and beta-blocker used to treat high blood pressure (hypertension). It works by relaxing blood vessels and slowing the heart rate, helping lower blood pressure. After a licensed provider reviews your prescription, your labetalol order ships from a licensed U.S. pharmacy.

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50-day supply · $0.30/tablet

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  1. Select your medication
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  3. Our licensed U.S. pharmacists fill your prescription
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Buy Labetalol 100mg (Trandate) Online

An alpha/beta-blocker for high blood pressure, including hypertension in pregnancy

Labetalol 100mg Quick Facts

Drug classAlpha/beta-adrenergic blocker
TreatsHigh blood pressure (hypertension)
FormTablet
Typical dosingTake 1 tablet by mouth twice daily.
Prescription requiredYes — prescription only

What Is Labetalol 100mg?

Labetalol is a prescription blood pressure medication that blocks both alpha and beta receptors. This dual action relaxes blood vessels and reduces the workload on the heart, which lowers blood pressure. Labetalol is FDA-approved to treat hypertension and may be used alone or with other blood pressure medicines. It is also commonly used by clinicians to manage high blood pressure during pregnancy.

What Does Labetalol 100mg Treat?

High blood pressure (hypertension)
Hypertension in combination with other antihypertensives
Hypertension during pregnancy (commonly used off-label per clinical guidelines)
Long-term blood pressure control to reduce cardiovascular risk

Labetalol 100mg Dosage

Initial: 100 mg by mouth twice daily.
Titrate: increase by 100 mg twice daily every 2–3 days as needed.
Maintenance: 200–400 mg by mouth twice daily.

Your prescriber will determine the dose and duration that are right for you. Always follow the directions on your prescription label.

Labetalol 100mg Side Effects

Common side effects

  • Dizziness
  • Fatigue
  • Nausea
  • Scalp tingling
  • Headache
  • Stuffy nose
  • Indigestion

Serious side effects

Stop taking this medication and seek medical attention right away if you experience:

  • Very slow heartbeat (bradycardia)
  • Fainting or severe lightheadedness (low blood pressure)
  • Difficulty breathing or wheezing (bronchospasm)
  • Signs of liver injury (jaundice, dark urine, severe fatigue)
  • Swelling of ankles or sudden weight gain (worsening heart failure)
  • Severe allergic reaction (rash, swelling, trouble breathing)

Warnings & Interactions

Do not use with asthma or obstructive airway disease
Contraindicated in severe bradycardia, heart block, or cardiogenic shock
Do not stop abruptly — taper under medical supervision
May cause liver injury; report symptoms promptly
Can mask signs of low blood sugar in diabetes
Use caution with other blood pressure medicines or calcium channel blockers
May cause dizziness when standing, especially early in treatment

Tell your prescriber about all medications, supplements, and health conditions before starting labetalol 100mg.

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Frequently Asked Questions

What is labetalol used for?

Labetalol is FDA-approved to treat high blood pressure (hypertension), either alone or with other blood pressure medicines. It is also widely used by clinicians to manage high blood pressure during pregnancy under medical supervision.

Do I need a prescription for labetalol?

Yes. Labetalol is a prescription-only medication in the United States. A licensed provider must review your health information and issue or verify a valid prescription before we can dispense it.

How does ordering and shipping work?

After you place your order, a licensed provider or pharmacist reviews your prescription and health details. Once approved, your medication is dispensed by our licensed U.S. pharmacy and shipped directly to your address.

How long does labetalol take to work?

Labetalol begins lowering blood pressure within hours of a dose, but it may take days to weeks of consistent use to see the full effect. Your provider may adjust your dose every few days until your blood pressure goal is reached.

Can I stop taking labetalol suddenly?

No. Stopping labetalol abruptly can cause a rebound rise in blood pressure or heart-related symptoms. Always taper the dose gradually under your provider's guidance.

Is labetalol safe during pregnancy?

Labetalol is one of the medications clinicians commonly use to manage high blood pressure in pregnancy. Only take it during pregnancy under the direction of your healthcare provider, who can weigh the benefits and risks for your situation.

What are the most common side effects of labetalol?

Common side effects include dizziness, fatigue, nausea, scalp tingling, and headache. Many effects lessen over time, but contact your provider if they persist or worsen.